5-Amino-1MQ
Inhibits NNMT → shifts methyl/NAD metabolism; proposed increase in adipocyte energy expenditure
AOD-9604
Lipolysis signaling via GH fragment without GH-mediated hyperglycemia
ARA-290
Innate-repair-receptor activation → neurovascular protection
BPC-157
Promotes angiogenesis, accelerates tissue regeneration, and protects gut integrity through growth-factor modulation
- Accelerated wound and tendon repair
- Gut healing and protection
- Vascular and nerve regeneration
- Anti-inflammatory effects
The gold standard for tissue repair across gut, musculoskeletal, vascular, and neural systems
Cartalax
Bioregulatory gene modulation in chondrocytes
CJC-1295
DAC-modified GHRH analog → extended half-life, sustained GH release amplification
DSIP
Delta-sleep inducing peptide → circadian rhythm modulation, stress-hormone regulation
Epitalon
Proposed epigenetic regulation of circadian rhythms; melatonin modulation
GHK-Cu
Copper-dependent collagen/elastin synthesis, MMP inhibition
- Dermal renewal and skin quality
- Connective-tissue strength
- Anti-inflammatory effects
Anti-aging crossover with tissue repair benefits
hGH
Direct GH supplementation → IGF-1 elevation, protein synthesis, lipolysis, tissue regeneration
- Enhanced muscle growth and recovery
- Fat loss and body recomposition
- Improved skin and connective tissue
- Bone density support
Requires careful dosing and monitoring; may suppress natural GH production
Ipamorelin
Selective ghrelin receptor agonist → GH pulse without cortisol/prolactin elevation
KPV
α-MSH fragment → NF-κB and cytokine suppression
- Calms inflammatory microenvironment
- Supports epithelial recovery
- Post-injury tissue repair
Potent anti-inflammatory for gut and systemic inflammation
L-Carnitine
Carnitine shuttle transports long-chain fatty acids into mitochondria for beta-oxidation
MOTS-C
Stress-responsive peptide that translocates to nucleus; up-regulates AMPK/FOXO programs
- Enhanced glucose and fatty-acid handling
- Improved exercise adaptation
- Metabolic flexibility enhancement
Weight recomposition support
NAD+
100-500mg
NAD+ is the prerequisite that makes all other healing possible. It transforms cellular metabolism from survival mode to repair mode.
- Transfer electrons for ATP production
- Power DNA repair
- Regulate gene expression
- Maintain cellular stress responses
Acting as a crucial electron carrier that powers the cell's energy-producing machinery.
Serving as a master regulator of cellular health by supporting enzymes like sirtuins and PARPs.
P21
CREB phosphorylation → BDNF transcription, dendritic spine growth, synaptic plasticity
Pinealon
CNS trophic claims; proposed oligopeptide regulatory effects on brain tissue
Retatrutide
Triple GLP-1 (satiety), GIP (insulinotropic/central effects), glucagon (lipolysis/EE) agonist
- Aggressive fat loss
- Enhanced energy expenditure
- Improved metabolic markers
- Requires resistance training 3×/week
Most aggressive metabolic intervention; must be paired with consistent resistance training
Semaglutide
GLP-1R agonism with albumin-binding for extended half-life
Semax
ACTH(4-10) analog → BDNF upregulation, D1/D2 receptor density increase, enkephalinase inhibition
- Enhanced focus and mental clarity
- Improved memory consolidation
- Neuroprotective effects
- Stress resilience and anxiety reduction
Powerful nootropic for CNS optimization, cognitive function, and stress response modulation
Selank
Tuftsin analog → GABAergic and serotonergic modulation, enkephalin stabilization
- Anxiety reduction without sedation
- Improved stress tolerance
- Enhanced mood stability
- Immune modulation
CNS, emotional regulation, and immune system support without sedative effects
Sermorelin
GHRH(1-29) analog → stimulates natural pulsatile GH release from pituitary
SS-31
Binds cardiolipin in inner mitochondrial membrane → stabilizes cristae, improves electron transport efficiency
- Reduced post-exertional malaise
- Improved HRV and orthostatic tolerance
- Enhanced mitochondrial function
- Steadier work output
Cardiolipin stabilization is dose-dependent early; tapering reduces cost while keeping membrane effects
TB-500
Actin polymerization → cell migration and angiogenesis
Tesamorelin
GHRH analog → pulsatile GH secretion, targeting visceral adipose tissue (VAT) reduction
- Visceral fat reduction
- Improved body composition
- Enhanced metabolic markers
- Lipid profile improvement
Targets growth hormone axis, metabolic function, and body composition optimization
Tirzepatide
GLP-1 satiety/gastric delay + GIP insulinotropic/central effects
VIP
Vasoactive Intestinal Peptide → immunomodulation, anti-inflammatory cytokine release, circadian regulation